Cyclobenzaprine: Uses, Side effects, dosage

Cyclobenzaprine is a muscle relaxer that relieves pain and discomfort caused by sprains, strains, and different muscle injuries.

  • It doesn’t directly act on the synapse or the muscle however relieves muscle spasms through a central action, probably at the brain stem level. cyclobenzaprine binds to the serotonin receptor and is taken into account a 5-HT2 receptor antagonist that reduces muscular tonus by decreasing the activity of descending serotonergic neurons.
  • The more common side effects of this drug will include: dizziness, drowsiness, dry mouth, fatigue, nausea, constipation, heartburn while Serious side effects may include ; Heart issues, and Serotonin syndrome.
  • The usual recommended dose of cyclobenzaprine dose is 15 or 30 mg once daily using extended release tablets or 5 or 10 mg 3 times daily using immediate release tablets .


  • Avoid if you’re allergic to that, or if you’ve got, congestive heart failure; a heart rhythm disorder, or you have recently had a heart attack; heart block; or a thyroid disorder.
  • Don’t take cyclobenzaprine if you have taken; monoamine oxidase inhibitor (MAOI) in the last two weeks. The combination of an monoamine oxidase inhibitor with cyclobenzaprine will turn out very serious, potentially serious side effects.
  • Cyclobenzaprine has been classified as pregnancy category B by the Food and Drug Administration. category B medication haven’t been shown to cause teratogenicity or fetal abnormalities in animal studies however usually haven’t been fully evaluated in humans. category B medication like cyclobenzaprine ought to be given throughout a pregnancy only if the physician determines that the risks are less than the advantages of the drug’s actions.
  • Take the incomprehensible dose as soon as you remember. Skip the missed dose if it’s nearly time for your next scheduled dose. don’t take further drugs to make up the missed dose.
  • Store at 25°C (77°F); excursions permissible to 15-30°C (59-86°F).

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